Publications

REISSIG, F., K. ZACHSLER, Z. NOVÝ, M. PETŘÍK, K. DVOŘÁKOVÁ BENDOVÁ, D. KURFÜRSTOVÁ, J. BOUCHAL, M. ĹUDIK, F. BRANDT, K. KOPKA, M. KHOYLOU, H. PIETZSCH, M. HAJDÚCH, C. MAMAT

Modulating the pharmacokinetic profile of Actinium-225-labeled macropa-derived radioconjugates by dual targeting of PSMA and albumin. Theranostics. 2022, 12(17), 7203-7215, ISSN: 1838-7640, PMID: 36438496,

BARUCIC, D., S. KAUSHIK, J. KYBIC, J. STANKOVÁ, P. DŽUBÁK, M. HAJDÚCH

Characterization of drug effects on cell cultures from phase-contrast microscopy images. Computers in Biology and Medicine. 2022, 151, 106171, ISSN: 0010-4825, PMID: 36306582,

BORKOVÁ, L., I. FRYDRYCH, B. VRÁNOVÁ, N. JAKUBCOVÁ, B. LIŠKOVÁ, P. DŽUBÁK, P. PAVLIŠ, M. HAJDÚCH, M. URBAN

Lupane derivatives containing various aryl substituents in the position 3 have selective cytostatic effect in leukemic cancer cells including resistant phenotypes. European Journal of Medicinal Chemistry. 2022, 244, 114850, ISSN: 0223-5234, PMID: 36283179,

YANG, C., L. POSTOVA SLAVETINSKA, M. FLEUTI, B. KLEPETAROVA, M. TICHÝ, S. GURSKÁ, P. PAVLIŠ, P. DŽUBÁK, M. HAJDÚCH, M. HOCEK

Synthesis of Polycyclic Hetero-Fused 7-Deazapurine Heterocycles and Nucleosides through C-H Dibenzothiophenation and Negishi Coupling. Journal of the American Chemical Society. 2022, 144(42), 19437-19446, ISSN: 0002-7863, PMID: 36245092,

ŘEZNÍČKOVÁ, E., S. KRAJČOVIČOVÁ, M. PERINA, A. KOVALOVA, M. SOURAL, V. KRYŠTOF

Modulation of FLT3-ITD and CDK9 in acute myeloid leukaemia cells by novel proteolysis targeting chimera (PROTAC). European Journal of Medicinal Chemistry. 2022, 243, 114792, ISSN: 0223-5234, PMID: 36191408, PDF.

HODOŇ, J., I. FRYDRYCH, Z. TRHLÍKOVÁ, J. POKORNÝ, L. BORKOVÁ, S. BENICKÁ, M. VLK, B. LIŠKOVÁ, A. KUBÍČKOVÁ, M. MEDVEDÍKOVÁ, M. PISÁR, J. ŠAREK, V. DAS, A. LIGASOVÁ, K. KOBERNA, P. DŽUBÁK, M. HAJDÚCH, M. URBAN

Triterpenoid pyrazines and pyridines - Synthesis, cytotoxicity, mechanism of action, preparation of prodrugs. European Journal of Medicinal Chemistry. 2022, 243, 114777, ISSN: 0223-5234, PMID: 36174412, PDF.

LEISCHNER FIALOVA, J., K. HONIGOVA, M. RAUDENSKA, L. MIKSATKOVA, R. ZOBALOVA, J. NAVRATIL, J. SMIGOVA, T. RAMJI MOTURU, T. VICAR, J. BALVAN, K. VESELA, N. ABRAMENKO, Z. KEJIK, R. KAPLANEK, J. GUMULEC, D. ROSEL, P. MARTASEK, J. BRABEK, M. JAKUBEK, J. NEUZIL, M. MASARIK

Pentamethinium salts suppress key metastatic processes by regulating mitochondrial function and inhibiting dihydroorotate dehydrogenase respiration. Biomedicine & Pharmacotherapy. 2022, 154, 113582, ISSN: 0753-3322, PMID: 36055111,

JORDA, R., L. HAVLÍČEK, M. PERINA, V. VOJÁČKOVÁ, T. POSPÍŠIL, S. DJUKIC, J. SKERLOVA, J. GRÚZ, N. RENESOVA, P. KLENER, P. ŘEZÁČOVÁ, M. STRNAD, V. KRYŠTOF

3,5,7-Substituted Pyrazolo[4,3- d]Pyrimidine Inhibitors of Cyclin-Dependent Kinases and Cyclin K Degraders. Journal of Medicinal Chemistry. 2022, 65(13), 8881-8896, ISSN: 0022-2623, PMID: 35749742,

SIKOROVÁ, K., S. MOON, H. YOON, A. STRNAD, J. SONG, M. PETŘEK

HLA class II variants defined by next generation sequencing are associated with sarcoidosis in Korean patients. Scientific Reports. 2022, 12(1), 9302, ISSN: 2045-2322, PMID: 35661780,

KLOS, D., M. DUŠEK, E. SAMOLOVA, M. ZATLOUKAL, V. NOZKOVA, N. NESNAS, L. PLACKOVA, R. KOPRNA, Z. SPISEK, H. VYLICILOVA, O. PLIHAL, K. DOLEZAL, J. VOLLER, A. KADLECOVA, M. STRNAD, L. PLÍHALOVÁ

New Water-Soluble Cytokinin Derivatives and Their Beneficial Impact on Barley Yield and Photosynthesis. Journal of Agricultural and Food Chemistry. 2022, 70(23), 7288-7301, ISSN: 0021-8561, PMID: 35658447,

Publications

Published in Top 10% journals in the field