Publications

Published in Top 10% journals in the field

ŘEHULKA, J., K. BÜRGLOVÁ, P. KREJČÍ, S. GURSKÁ, P. HRADIL, M. HAJDÚCH, P. DŽUBÁK, J. HLAVÁČ
Fluorinated derivatives of 2-phenyl-3-hydroxy-4(1H)-quinolinone as tubulin polymerization inhibitors. European Journal of Medicinal Chemistry. 2020, 192, 112176, ISSN: 0223-5234, PMID: 32120327,
SAID, M., W. ELDEHNA, A. NOCENTINI, S. FAHIM, A. BONARDI, A. ELGAZAR, V. KRYŠTOF, D. SOLIMAN, H. ABDEL-AZIZ, P. GRATTERI, S. ABOU-SERI, C. SUPURAN
Sulfonamide-based ring-fused analogues for CAN508 as novel carbonic anhydrase inhibitors endowed with antitumor activity: Design, synthesis, and in vitro biological evaluation. European Journal of Medicinal Chemistry. 2020, 189(2020), 112019, ISSN: 0223-5234, PMID: 31972394,
JORDA, R., P. MAGAR, D. HENDRYCHOVA, K. PAUK, M. DIBUS, E. PILAROVA, A. IMRAMOVSKY, V. KRYŠTOF
Novel modified leucine and phenylalanine dipeptides modulate viability and attachment of cancer cells. European Journal of Medicinal Chemistry. 2020, 188, 112036, ISSN: 0223-5234, PMID: 31931341,
BORKOVÁ, L., I. FRYDRYCH, N. JAKUBCOVÁ, R. ADÁMEK, B. LIŠKOVÁ, S. GURSKÁ, M. MEDVEDÍKOVÁ, M. HAJDÚCH, M. URBAN
Synthesis and biological evaluation of triterpenoid thiazoles derived from betulonic acid, dihydrobetulonic acid, and ursonic acid. European Journal of Medicinal Chemistry. 2019, 185, 111806, ISSN: 0223-5234, PMID: 31677446,
GRUNER, B., J. BRYNDA, V. DAS, V. SICHA, J. ŠTĚPÁNKOVÁ, J. NEKVINDA, J. HOLUB, K. POSPISILOVA, M. FABRY, P. PACHL, V. KRAL, M. KUGLER, V. MAŠEK, M. MEDVEDÍKOVÁ, S. MATEJKOVA, A. NOVÁ, B. LIŠKOVÁ, S. GURSKÁ, P. DŽUBÁK, M. HAJDÚCH, P. ŘEZÁČOVÁ
Metallacarborane Sulfamides: Unconventional, Specific, and Highly Selective Inhibitors of Carbonic Anhydrase IX. Journal of Medicinal Chemistry. 2019, 62(21), 9560-9575, ISSN: 0022-2623, PMID: 31568723,
HODOŇ, J., L. BORKOVÁ, J. POKORNÝ, A. KAZAKOVA, M. URBAN
Design and synthesis of pentacyclic triterpene conjugates and their use in medicinal research. European Journal of Medicinal Chemistry. 2019, 182, 111653, ISSN: 0223-5234, PMID: 31499360,
KADLECOVA, A., B. MAKOVA, M. ARTAL-SANZ, M. STRNAD, J. VOLLER
The plant hormone kinetin in disease therapy and healthy aging. Ageing Rsearch Reviews. 2019, 55, 100958, ISSN: 1568-1637, PMID: 31479763,
VANZO, R., J. BARTKOVA, J. MERCHUT-MAYA, A. HALL., J. BOUCHAL, L. DYRSKJOT, L. FRANKEL, V. GORGOULIS, A. MAYA-MENDOZA, M. JAATTELA, J. BÁRTEK
Autophagy role(s) in response to oncogenes and DNA replication stress. Cell Death and Differentiation. 2019, 27(3), 1134-1153, ISSN: 1350-9047, PMID: 31409894,
VANDA, D., P. ZAJDEL, M. SOURAL
Imidazopyridine-based selective and multifunctional ligands of biological targets associated with psychiatric and neurodegenerative diseases. European Journal of Medicinal Chemistry. 2019, 181, 111569, ISSN: 0223-5234, PMID: 31404862,
VOUGAS, K., T. SAKELAROPOULOS, A. KOTSINAS, G. FOUKAS, A. NTARGARAS, F. KOINIS, A. POLYZOS, V. MYRIANTHOPOULOS, H. ZHOU, S. NARANG, V. GEORGOULIAS, L. ALEXOPOULOS, I. AIFANTIS, P. TOWNSEND, P. SFIKAKIS, R. FITZGERALD, D. THANOS, J. BÁRTEK, R. PETTY, A. TSIRIGOS, V. GORGOULIS
Machine learning and data mining frameworks for predicting drug response in cancer: An overview and a novel in silico screening process based on association rule mining. Pharmacology & Therapeutics. 2019, 203, 107395, ISSN: 0163-7258, PMID: 31374225,