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Publications

Published in Top 10% journals in the field

ŠKROTT, Z., M. MISTRÍK, K. ANDERSEN, S. FRIIS, D. MAJERA, J. GURSKÝ, T. OŽDIAN, J. BARTKOVA, Z. TURI, P. MOUDRÝ, M. KRAUS, M. MEDVEDÍKOVÁ, J. VÁCLAVKOVÁ, P. DŽUBÁK, I. VROBEL, P. POUCKOVA, J. SEDLACEK, A. MIKLOVICOVA, A. KUTT, J. MATTOVA, C. DRIESSEN, Q. DOU, J. OLSEN, M. HAJDÚCH, B. CVEK, R. DESHAIES, J. BÁRTEK
Alcohol-abuse drug disulfiram targets cancer via p97 segregase adaptor NPL4. Nature. 2017, 552(7684), 194-199, ISSN: 0028-0836, PMID: 29211715,
MODER, M., G. VELIMEZI, M. OWUSU, A. MAZOUZI, M. WIEDNER, J. FERREIRA DA SILVA, L. ROBINSON-GARCIA, F. SCHISCHLIK, R. SLAVKOVSKÝ, R. KRALOVICS, B. SCHUSTER, C. BOCK, T. IDEKER, S. JACKSON, J. MENCHE, J. LOIZOU
Parallel genome-wide screens identify synthetic viable interactions between the BLM helicase complex and Fanconi anemia. Nature Communications. 2017, 8(1), 1238, ISSN: 2041-1723, PMID: 29089570,
EIGNEROVA, B., M. TICHÝ, J. KRASULOVA, L. RÁROVÁ, R. CHRISTOVÁ, M. URBAN, B. BEDNARCZYK-CWYNAR, M. HAJDÚCH, J. ŠAREK
Q1_Synthesis and antiproliferative properties of new hydrophilic esters of triterpenic acids. European Journal of Medicinal Chemistry. 2017, 140, 403-420, ISSN: 0223-5234, PMID: 28987603,
KARLÍKOVÁ, R., K. MIČOVÁ, L. NAJDEKR, A. GARDLO, T. ADAM, P. MAJEROVÁ, D. FRIEDECKÝ, A. KOVAC
Metabolic status of CSF distinguishes rats with tauopathy from controls. Alzheimer's Research & Therapy. 2017, 9(1), 78, ISSN: 1758-9193, PMID: 28934963,
VRZALIKOVA, K., M. IBRAHIM, M. VOCKERODT, T. PERRY, S. MARGIELEWSKA, L. LUPINO, E. NAGY, E. SOILLEUX, D. LIEBELT, R. HOLLOWS, A. LAST, G. REYNOLDS, M. ABDULLAH, H. CURLEY, M. CARE, D. KRAPPMANN, R. TOOZE, J. ALLEGOOD, S. SPIEGEL, W. WEI, C. WOODMAN, P. MURRAY
S1PR1 drives a feed forward signalling loop to regulate BATF3 and the transcriptional programme of Hodgkin lymphoma cells. Leukemia. 2018, 32(1), 214-223, ISSN: 0887-6924, PMID: 28878352,
EFFENBERG, R., P. TURANEK KNOTIGOVA, D. ZYKA, H. CELECHOVSKA, J. MASEK, E. BARTHELDYOVA, F. HUBATKA, S. KOUDELKA, R. LUKAC, A. KOVALOVA, D. SAMAN, M. KŘUPKA, L. BARKOCZIOVA, P. KOSZTYU, M. ŠEBELA, L. DROZ, M. HUCKO, M. KANASKOVA, A. MILLER, M. RAŠKA, M. LEDVINA, J. TURANEK
Nonpyrogenic Molecular Adjuvants Based on norAbu-Muramyldipeptide and norAbu-Glucosaminyl Muramyldipeptide: Synthesis, Molecular Mechanisms of Action, and Biological Activities in Vitro and in Vivo. Journal of Medicinal Chemistry. 2017, 60(18), 7745-7763, ISSN: 0022-2623, PMID: 28829599,
NARDONE, G., J. OLIVER-DE LA CRUZ, J. VRBSKY, C. MARTINI, J. PRIBYL, P. SKLADAL, M. PESL, G. CALUORI, S. PAGLIARI, F. MARTINO, Z. MACEČKOVÁ, M. HAJDÚCH, A. SANZ-GARCIA, N. PUGNO, G. STOKIN, G. FORTE
YAP regulates cell mechanics by controlling focal adhesion assembly. Nature Communications. 2017, 15, 8:15321, ISSN: 2041-1723, PMID: 28504269,
VAN GOOL, A., F. BIETRIX, E. CALDENHOVEN, K. ZATLOUKAL, A. SCHERER, J. LITTON, G. MEIJER, N. BLOMBERG, A. SMITH, B. MONS, J. HERINGA, W. KOOT, M. SMIT, M. HAJDÚCH, T. RIJNDERS, A. USSI
Bridging the translational innovation gap through good biomarker practice. Nature Reviews. Drug Discovery. 2017, 16(9), 587-588, ISSN: 1474-1776, PMID: 28450744,
TICHÝ, M., S. SMOLEN, E. TLOUŠŤOVÁ, R. POHL, T. OŽDIAN, K. HEJTMÁNKOVÁ, B. LIŠKOVÁ, S. GURSKÁ, P. DŽUBÁK, M. HAJDÚCH, M. HOCEK
Synthesis and Cytostatic and Antiviral Profiling of Thieno-Fused 7-Deazapurine Ribonucleosides. Journal of Medicinal Chemistry. 2017, 60(6), 2411-2424, ISSN: 0022-2623, PMID: 28221790,
CHROMÁ, K., M. MISTRÍK, P. MOUDRÝ, J. GURSKÝ, M. LIPTAY, R. STRAUSS, Z. ŠKROTT, R. VRTEL, J. BARTKOVA, J. KRAMARA, J. BÁRTEK
Tumors overexpressing RNF168 show altered DNA repair and responses to genotoxic treatments, genomic instability and resistance to proteotoxic stress. Oncogene. 2017, 36(17), 2405-2422, ISSN: 0950-9232, PMID: 27841863,